Compile Data Set for Download or QSAR
Found 11 of ic50 data for polymerid = 50004846
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))TBA
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 69.6nMAssay Description:Inhibition of human SGK3 using GRPRTSSFAEG as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5KB8PubMed
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))TBA
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 76.5nMAssay Description:Inhibition of human SGK3 using GRPRTSSFAEG as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W380MTPubMed
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))TBA
LigandPNGBDBM269003(N-[4-(3-Amino-1H-pyrazolo[3,4-d]pyrimidin-6-yl)-ph...)copy SMILEScopy InChI
Affinity DataIC50: 211nMAssay Description:Inhibition of human SGK3 in presence 500 uM presence of ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P55SCWPubMed
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))TBA
LigandPNGBDBM50462709(CHEMBL4245507)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of SGK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XP77MHPubMed
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))TBA
LigandPNGBDBM50443628(CHEMBL3092468 | US9174993, 35 | US9221828, 35)copy SMILEScopy InChI
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of human SGK3 in presence of 500 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28S4RJTPubMed
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))TBA
LigandPNGBDBM50429867(CHEMBL2333365)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of SGK3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC847XPubMed
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))TBA
LigandPNGBDBM50519662(CHEMBL4438748)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human SGK3 (119 to end residues) using GRPRTSSFAEGKK as substrate incubated for 40 mins in presence of [gamma33P]ATP by rad...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC93FGPubMed
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))TBA
LigandPNGBDBM50135286(CHEMBL3745885)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human SGK3 using [GRPRTSSFAEG] as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24Q7WT8PubMed
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))TBA
LigandPNGBDBM50443636(CHEMBL3092460 | US9174993, 1 | US9221828, 1)copy SMILEScopy InChI
Affinity DataIC50: 2.33E+4nMAssay Description:Inhibition of human SGK3 in presence of 500 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28S4RJTPubMed
TargetSerine/threonine-protein kinase Sgk3(Homo sapiens (Human))TBA
LigandPNGBDBM50537742(CHEMBL4634634 | US11179389, Compound 1-14)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against cytosolic c-SrcMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed